[The tartrate salt form of tolterodine, a benzhydryl compound and a muscarinic receptor antagonist possessing both antimuscarinic and antispasmodic properties. Both tolterodine and its active metabolite, 5-hydroxymethyltolterodine, competitively blocks muscarinic receptors, thereby inhibiting acetylcholine receptor binding. This antagonistic action results in an increase in residual urine, reflecting an incomplete emptying of the bladder, and a decrease in detrusor pressure, indicating an antimuscarinic action on the lower urinary tract.. The 5-hydroxymethyl metabolite appears to contribute significantly to the therapeutic effects. ( NCI )]
UMLS (NCI) C0724710TOLTERODINE TARTRATE PREPARATION
- Organic Chemical
- Pharmacologic Substance
Relation/PAR: Tolterodine
Relation/CHD: TOLTERODINE TARTRATE 1 MG
TOLTERODINE TARTRATE 2 MG
TOLTERODINE TARTRATE 4 MG